Development of β-lactoglobulin-specific chimeric human IgEκ monoclonal antibodies for in vitro safety assessment of whey hydrolysates

PLoS One. 2014 Aug 25;9(8):e106025. doi: 10.1371/journal.pone.0106025. eCollection 2014.

Abstract

Background: Cow's milk-derived whey hydrolysates are nutritional substitutes for allergic infants. Safety or residual allergenicity assessment of these whey hydrolysates is crucial. Currently, rat basophilic leukemia RBL-2H3 cells expressing the human IgE receptor α-chain (huFcεRIα-RBL-2H3), sensitized with serum IgE from cow's milk allergic children, are being employed to assess in vitro residual allergenicity of these whey hydrolysates. However, limited availability and inter-lot variation of these allergic sera impede standardization of whey hydrolysate safety testing in degranulation assays.

Objective: An oligoclonal pool of chimeric human (chu)IgE antibodies against bovine β-lactoglobulin (a major allergen in whey) was generated to increase sensitivity, specificity, and reproducibility of existing degranulation assays.

Methods: Mice were immunized with bovine β-lactoglobulin, and subsequently the variable domains of dissimilar anti-β-lactoglobulin mouse IgG antibodies were cloned and sequenced. Six chimeric antibodies were generated comprising mouse variable domains and human constant IgE/κ domains.

Results: After sensitization with this pool of anti-β-lactoglobulin chuIgEs, huFcεRIα-expressing RBL-2H3 cells demonstrated degranulation upon cross-linking with whey, native 18 kDa β-lactoglobulin, and 5-10 kDa whey hydrolysates, whereas a 3 kDa whey hydrolysate and cow's milk powder (mainly casein) showed no degranulation. In parallel, allergic serum IgEs were less sensitive. In addition, our pool anti-β-lactoglobulin chuIgEs recognized multiple allergenic immunodominant regions on β-lactoglobulin, which were also recognized by serum IgEs from cow's milk allergic children.

Conclusion: Usage of our 'unlimited' source and well-defined pool of β-lactoglobulin-specific recombinant chuIgEs to sensitize huFcεRIα on RBL-2H3 cells showed to be a relevant and sensitive alternative for serum IgEs from cow's milk allergic patients to assess safety of whey-based non-allergic hydrolyzed formula.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Allergens / immunology
  • Animals
  • Antibodies, Monoclonal / immunology*
  • Caseins / immunology
  • Cattle
  • Cell Line
  • Child
  • Female
  • Humans
  • Immunoglobulin E / immunology*
  • Lactoglobulins / immunology*
  • Mice
  • Mice, Inbred BALB C
  • Milk Hypersensitivity / immunology
  • Protein Hydrolysates / immunology
  • Rats
  • Receptors, IgE / immunology
  • Reproducibility of Results
  • Whey / immunology*
  • Whey Proteins / immunology

Substances

  • Allergens
  • Antibodies, Monoclonal
  • Caseins
  • FCER1A protein, human
  • Lactoglobulins
  • Protein Hydrolysates
  • Receptors, IgE
  • Whey Proteins
  • Immunoglobulin E

Grants and funding

This study is financially supported by Agentschap NL within the SLIM (SneLler van Innovatie naar Mens) project in frame of 'Pieken in de Delta' (PID 101063) to improve fast implementation of alternatives for animal testing. Funding received by KK, PS, LBS, LC, MdH, NdJ, JG, LB and LK. The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.