DNA replication-dependent induction of gene proximity by androgen

Hum Mol Genet. 2015 Feb 15;24(4):963-71. doi: 10.1093/hmg/ddu508. Epub 2014 Oct 3.

Abstract

The male hormone androgen, working through the androgen receptor (AR), plays a major role in physiological process and disease development. Previous studies of AR mainly focus on its transcriptional activity. Here, we found that androgen-induced TMPRSS2 and ERG gene proximity is mediated by AR control of DNA replication rather than gene transcription. We demonstrate that, in both AR transactivation-positive and -negative prostate cells, androgen regulates DNA replication and androgen-induced gene proximity relies on both DNA replication-licensing and actual DNA replication activity. Androgen stimulation advances DNA replication timing of certain genomic regions, which may potentially increase gene proximity through sharing the same replication factory at a similar time. Therefore, we have revealed novel mechanisms of AR biological function, which will stimulate new research directions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Androgens / metabolism*
  • Androgens / pharmacology
  • Cell Line
  • DNA Replication*
  • Dihydrotestosterone / metabolism
  • Dihydrotestosterone / pharmacology
  • Gene Expression Regulation* / drug effects
  • Humans
  • Male
  • Receptors, Androgen / metabolism
  • Serine Endopeptidases / genetics
  • Trans-Activators / genetics
  • Transcriptional Activation* / drug effects
  • Transcriptional Regulator ERG

Substances

  • Androgens
  • ERG protein, human
  • Receptors, Androgen
  • Trans-Activators
  • Transcriptional Regulator ERG
  • Dihydrotestosterone
  • Serine Endopeptidases
  • TMPRSS2 protein, human