Dermatological approach to vemurafenib skin toxicity: a single centre experience

G Ital Dermatol Venereol. 2016 Feb;151(1):25-31. Epub 2014 Oct 9.

Abstract

Background: Targeted therapies have recently changed the approach to advanced melanoma. RAF inhibitors represent the emerging standard of care for metastatic BRAF mutated melanomas. Cutaneous reactions are the most common side effects during vemurafenib treatment, and affect the quality of life. The aim of this study was to provide some practical advices to manage the drug related cutaneous reactions.

Methods: A cohort of BRAF-mutated metastatic melanoma patients treated at our institution included 20 female and 21 male patients; median age was 56 years (32-87 years). All patients were treated at a dose of 960 mg b.i.d. orally.

Results: After a median treatment duration of 7 months (range 0.5-25.2), 29/39 patients (74.4%) developed cutaneous toxicities. We identified 22 cases of maculo-papular rash (56%) and 18 of warts (46%); in a total of 10 cases we observed alterations of keratinization (25.6%), while 6 of our patients presented photosensitivity (15 %). Six patients developed keratoacanthomas; no second melanomas were observed.

Conclusions: Skin involvement during vemurafenib treatment is frequent but in the majority of cases cutaneous side effects are self-limiting and easy to manage. Moreover, sun protection is mandatory in vemurafenib treated patients, and should be started together with BRAF inhibitor in order to minimize the impact of photosensitivity on quality of life.

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Aged, 80 and over
  • Antineoplastic Agents / administration & dosage*
  • Antineoplastic Agents / adverse effects
  • Biomarkers, Tumor / genetics
  • Dose-Response Relationship, Drug
  • Exanthema / etiology
  • Female
  • Humans
  • Indoles / administration & dosage*
  • Indoles / adverse effects
  • Keratinocytes / drug effects
  • Keratoacanthoma / chemically induced*
  • Male
  • Melanoma / drug therapy*
  • Melanoma / pathology
  • Melanoma, Cutaneous Malignant
  • Middle Aged
  • Molecular Targeted Therapy / adverse effects
  • Mutation
  • Photosensitivity Disorders / chemically induced*
  • Proto-Oncogene Proteins B-raf / genetics
  • Risk Factors
  • Skin Neoplasms / drug therapy*
  • Skin Neoplasms / pathology
  • Sulfonamides / administration & dosage*
  • Sulfonamides / adverse effects
  • Vemurafenib
  • Warts / chemically induced

Substances

  • Antineoplastic Agents
  • Biomarkers, Tumor
  • Indoles
  • Sulfonamides
  • Vemurafenib
  • BRAF protein, human
  • Proto-Oncogene Proteins B-raf