αB-crystallin interacts with and prevents stress-activated proteolysis of focal adhesion kinase by calpain in cardiomyocytes

Nat Commun. 2014 Oct 16:5:5159. doi: 10.1038/ncomms6159.

Abstract

Focal adhesion kinase (FAK) contributes to cellular homeostasis under stress conditions. Here we show that αB-crystallin interacts with and confers protection to FAK against calpain-mediated proteolysis in cardiomyocytes. A hydrophobic patch mapped between helices 1 and 4 of the FAK FAT domain was found to bind to the β4-β8 groove of αB-crystallin. Such an interaction requires FAK tyrosine 925 and is enhanced following its phosphorylation by Src, which occurs upon FAK stimulation. αB-crystallin silencing results in calpain-dependent FAK depletion and in the increased apoptosis of cardiomyocytes in response to mechanical stress. FAK overexpression protects cardiomyocytes depleted of αB-crystallin against the stretch-induced apoptosis. Consistently, load-induced apoptosis is blunted in the hearts from cardiac-specific FAK transgenic mice transiently depleted of αB-crystallin by RNA interference. These studies define a role for αB-crystallin in controlling FAK function and cardiomyocyte survival through the prevention of calpain-mediated degradation of FAK.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Aorta / metabolism
  • Apoptosis
  • Calpain / metabolism*
  • Cell Survival
  • Fluorescence Resonance Energy Transfer
  • Focal Adhesion Protein-Tyrosine Kinases / metabolism*
  • Gene Expression Regulation, Enzymologic*
  • Gene Silencing
  • Homeostasis
  • Male
  • Mice
  • Mice, Transgenic
  • Microscopy, Fluorescence
  • Models, Molecular
  • Myocardium / metabolism
  • Myocytes, Cardiac / cytology*
  • Phosphorylation
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Rats
  • Rats, Wistar
  • Stress, Mechanical
  • alpha-Crystallin B Chain / chemistry*
  • src-Family Kinases / metabolism

Substances

  • alpha-Crystallin B Chain
  • Focal Adhesion Protein-Tyrosine Kinases
  • src-Family Kinases
  • Calpain