Ligand selectivity in stabilising tandem parallel folded G-quadruplex motifs in human telomeric DNA sequences

Chem Commun (Camb). 2014 Dec 14;50(96):15202-5. doi: 10.1039/c4cc07487d.

Abstract

Biophysical studies of ligand interactions with three human telomeric repeat sequences (d(AGGG(TTAGGG)n, n = 3, 7 and 11)) show that an oxazole-based 'click' ligand, which induces parallel folded quadruplexes, preferentially stabilises longer telomeric repeats providing evidence for selectivity in binding at the interface between tandem quadruplex motifs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Base Sequence
  • Binding Sites
  • Circular Dichroism
  • Click Chemistry
  • G-Quadruplexes*
  • Humans
  • Ligands*
  • Molecular Dynamics Simulation
  • Nucleic Acid Conformation
  • Oxazoles / chemistry
  • Telomere / chemistry*

Substances

  • Ligands
  • Oxazoles