Soluble or soluble/membrane TNF-α inhibitors protect the brain from focal ischemic injury in rats

Int J Neurosci. 2015;125(12):936-40. doi: 10.3109/00207454.2014.980906. Epub 2014 Nov 25.

Abstract

Tumor Necrosis Factor-alpha (TNF-α) is an immunomodulatory and proinflammatory cytokine implicated in neuro-inflammation and neuronal damage in response to cerebral ischemia. The present study tested the hypothesis that anti-TNF-α agents may be protective against cerebral infarction. Transient focal ischemia was artificially induced in anesthetized adult male Wistar rats (300-350 g) by middle cerebral artery occlusion (MCAO) with an intraluminal suture. TNF-α function was interfered with either a chimeric monoclonal antibody against TNF-α (infliximab-7 mg/kg) aiming to TNF-α soluble and membrane-attached form; or a chimeric fusion protein of TNF-α receptor-2 with a fragment crystallizable (Fc) region of IgG1 (etanercept-5 mg/kg) aiming for the TNF-α soluble form. Both agents were administered intraperitoneally 0 or 6 h after inducing ischemia. Infarct volume was measured by 2,3,5-triphenyltetrazolium chloride staining. Cerebral infarct volume was significantly reduced in either etanercept or infliximab-treated group compared with non-treated MCAO rats 24 h after reperfusion. These results suggest that anti-TNF-α agents may reduce focal ischemic injury in rats.

Keywords: anti TNF-α; brain ischemia; etanercept; experimental brain research; infliximab.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain Infarction / etiology
  • Brain Infarction / prevention & control
  • Brain Injuries / etiology
  • Brain Injuries / prevention & control*
  • Disease Models, Animal
  • Etanercept / therapeutic use*
  • Infarction, Middle Cerebral Artery / complications
  • Infarction, Middle Cerebral Artery / drug therapy
  • Infliximab / therapeutic use*
  • Male
  • Neuroprotective Agents / therapeutic use*
  • Rats
  • Rats, Wistar
  • Time Factors
  • Tumor Necrosis Factor-alpha / immunology
  • Tumor Necrosis Factor-alpha / metabolism*

Substances

  • Neuroprotective Agents
  • Tumor Necrosis Factor-alpha
  • Infliximab
  • Etanercept