Inhibitory effects of C-type natriuretic peptide on the differentiation of cardiac fibroblasts, and secretion of monocyte chemoattractant protein-1 and plasminogen activator inhibitor-1

Mol Med Rep. 2015 Jan;11(1):159-65. doi: 10.3892/mmr.2014.2763. Epub 2014 Oct 23.

Abstract

The present study aimed to investigate the effect of C-type natriuretic peptide (CNP) on the function of cardiac fibroblasts (CFs). Western blotting was used to investigate the expression of myofibroblast marker proteins: α-smooth muscle actin (α-SMA), extra domain-A fibronectin, collagen I and collagen III, and the activity of extracellular signal-regulated kinase 1/2 (ERK1/2). Immunofluorescence was used to examine the morphological changes; a transwell assay was used to analyze migration, and reverse transcription-quantitative polymerase chain reaction and ELISA were employed to determine the mRNA expression and protein secretion of monocyte chemoattractant protein-1 (MCP-1) and plasminogen activator inhibitor-1 (PAI-1). The results demonstrated that CNP significantly reduced the protein expression of α-SMA, fibronectin, collagen I and collagen III, and suppressed the migratory ability of CFs. Additionally, the mRNA and protein expression of MCP-1 and PAI-1 was inhibited under the CNP treatment; and this effect was mediated by the inhibition of the ERK1/2 activity. In conclusion, CNP inhibited cardiac fibroblast differentiation and migration, and reduced the secretion of MCP-1 and PAI-1, which demonstrates novel mechanisms to explain the antifibrotic effect of CNP.

MeSH terms

  • Animals
  • Animals, Newborn
  • Cell Differentiation / drug effects*
  • Cell Movement / drug effects
  • Chemokine CCL2 / genetics
  • Chemokine CCL2 / metabolism*
  • Enzyme Activation / drug effects
  • Gene Expression
  • Mitogen-Activated Protein Kinase 1 / metabolism
  • Mitogen-Activated Protein Kinase 3 / metabolism
  • Myoblasts, Cardiac / cytology*
  • Myoblasts, Cardiac / metabolism*
  • Myofibroblasts / cytology*
  • Myofibroblasts / metabolism*
  • Natriuretic Peptide, C-Type / pharmacology*
  • Plasminogen Activator Inhibitor 1 / genetics
  • Plasminogen Activator Inhibitor 1 / metabolism*
  • Primary Cell Culture
  • Rats

Substances

  • Chemokine CCL2
  • Plasminogen Activator Inhibitor 1
  • Natriuretic Peptide, C-Type
  • Mitogen-Activated Protein Kinase 1
  • Mitogen-Activated Protein Kinase 3