[Pharmacological characteristics of glycine receptors in rat hippocampal pyramidal cells]

Zhong Nan Da Xue Xue Bao Yi Xue Ban. 2014 Oct;39(10):989-93. doi: 10.11817/j.issn.1672-7347.2014.10.001.
[Article in Chinese]

Abstract

Objective: To investigate function of glycine receptors (GlyRs) at the hippocampal CA1 pyramidal cells and to characterize the pharmacological properties of these receptors at early postnatal stage.

Methods: We used whole cell patch clamp recording to study the current response in the acutely prepared hippocampal slices from postnatal day 11-13 rats induced by glycine applied in the artificial cerebrospinal fluid.

Results: Application of glycine to the pyramidal cells elicited strychnine sensitive chloride currents. EC50 for GlyRs respond to glycine was 123. 23 μmol/L and Hill coefficient was 1.24. Picrotoxin could partly blocked the currents.

Conclusion: Strychnine sensitive glycine receptors are functionally expressed in CA1 pyramidal neurons in rat hippocampal CA1 area at early postnatal stage, and some of GlyRs are αβ heteromeric receptors.

MeSH terms

  • Animals
  • CA1 Region, Hippocampal / cytology*
  • Glycine / pharmacology
  • Patch-Clamp Techniques
  • Pyramidal Cells / drug effects*
  • Rats
  • Receptors, Glycine / metabolism*
  • Strychnine / pharmacology

Substances

  • Receptors, Glycine
  • Strychnine
  • Glycine