Oxidized low-density lipoprotein inhibits THP-1-derived macrophage autophagy via TET2 down-regulation

Lipids. 2015 Feb;50(2):177-83. doi: 10.1007/s11745-014-3977-5. Epub 2014 Dec 14.

Abstract

Oxidized low-density lipoprotein (ox-LDL) is an independent risk factor of atherosclerosis. However, the mechanism underlying its pro-atherosclerosis roles has not yet been well explored. DNA demethylation modification, via DNA methyltransferases or ten-eleven-translocation (TET) family, is a crisis epigenetic regulation for various biological and pathological processes. This study aimed to investigate the effects of ox-LDL on macrophage autophagy and its potential epigenetic mechanism. Results showed that after treatment with 0, 10, 20, 40 or 80 mg/L ox-LDL for 24 h, the autophagy markers Beclin 1 and LC3 expression were obviously decreased at protein levels (P < 0.05). The mRNA and protein expression of TET2 was evidently decreased (P < 0.05). After pre-treatment with TET2 siRNA, the mRNA and protein levels of Beclin 1 and LC3 decreased compared with the 80 mg/L treatment group (P < 0.01). The mRNA and protein levels of Beclin 1 and LC3-II were up-regulated (P < 0.05) in the 5-aza-2'-deoxycytidine (a DNA methyltransferase inhibitor) of pretreatment group. Consistent with the Western blot results, cell immunofluorescence showed that the protein concentration of LC3-II decreased in the TET2 siRNA group and increased in the 5-aza-2'-deoxycytidine group. Taken together, these results showed that DNA demethylation modifications regulate ox-LDL-treated THP-1 macrophages autophagy and TET2 might be a novel regulator.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis Regulatory Proteins / genetics
  • Autophagy*
  • Beclin-1
  • Cell Line
  • DNA-Binding Proteins / genetics*
  • Dioxygenases
  • Down-Regulation*
  • Epigenesis, Genetic
  • Humans
  • Lipoproteins, LDL / metabolism*
  • Macrophages / cytology*
  • Macrophages / metabolism
  • Membrane Proteins / genetics
  • Microtubule-Associated Proteins / genetics
  • Proto-Oncogene Proteins / genetics*
  • RNA Interference
  • RNA, Small Interfering / genetics

Substances

  • Apoptosis Regulatory Proteins
  • BECN1 protein, human
  • Beclin-1
  • DNA-Binding Proteins
  • Lipoproteins, LDL
  • MAP1LC3A protein, human
  • Membrane Proteins
  • Microtubule-Associated Proteins
  • Proto-Oncogene Proteins
  • RNA, Small Interfering
  • oxidized low density lipoprotein
  • Dioxygenases
  • TET2 protein, human