[Inhibition of sunitinib on the expressions of PD-L1 and PD-L2 of mouse bone marrow-derived dendritic cells]

Xi Bao Yu Fen Zi Mian Yi Xue Za Zhi. 2015 Jan;31(1):10-3.
[Article in Chinese]

Abstract

Objective: To observe the changes of programmed death-1 ligand 1 (PD-L1) and PD-L2 expressions on mouse bone marrow-derived dendritic cells (DCs) stimulated by sunitinib.

Methods: DCs were randomly divided into four groups which were treated with sunitinib (100, 200, 300 ng/mL) and dimethylsulfoxide (DMSO), respectively. After 48 hours, PD-L1 and PD-L2 expression levels were analyzed by flow cytometry.

Results: Compared with the control group, the expression of PD-L1 on mature DCs (mDCs) and all DCs [including mature DCs and immature DCs (imDCs)] was significantly down-regulated in sunitinib treatment groups. The PD-L1 expression percentages of imDCs, mDCs and DCs were significantly reduced in sunitinib treatment groups; the percentage of mDCs expressing PD-L2 also dropped in all treatment groups, and the percentage of DCs expressing PD-L2 decreased in 100 and 300 ng/mL sunitinib treatment groups.

Conclusion: Sunitinib can significantly reduce the expressions of PD-L1 and PD-L2 on mouse DCs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology*
  • B7-H1 Antigen / genetics*
  • B7-H1 Antigen / metabolism
  • Bone Marrow / drug effects*
  • Bone Marrow / metabolism
  • Cells, Cultured
  • Dendritic Cells / drug effects*
  • Dendritic Cells / metabolism
  • Female
  • Gene Expression / drug effects
  • Indoles / pharmacology*
  • Mice
  • Mice, Inbred C57BL
  • Programmed Cell Death 1 Ligand 2 Protein / genetics*
  • Programmed Cell Death 1 Ligand 2 Protein / metabolism
  • Pyrroles / pharmacology*
  • Sunitinib

Substances

  • Antineoplastic Agents
  • B7-H1 Antigen
  • Cd274 protein, mouse
  • Indoles
  • Pdcd1lg2 protein, mouse
  • Programmed Cell Death 1 Ligand 2 Protein
  • Pyrroles
  • Sunitinib