[ERKl/2 signaling pathway mediates heme oxygenase-1 up-regulation by minocycline in PC12 cells exposed to oxygen glucose deprivation]

Nan Fang Yi Ke Da Xue Xue Bao. 2015 Jan;35(1):117-20.
[Article in Chinese]

Abstract

Objective: To investigate the effects of minocycline in promoting the survival of pheochromocytoma (PCI2) cells exposed to oxygen glucose deprivation (OGD) and explore the underlying mechanisms.

Methods: An in vitro cell model of cerebral ischemia was established by OGD for 6 h in PCI2 cells with pretreatment with minocycline or an ERK1/2 inhibitor. At 24 h after OGD injury, the cells were evaluated for cell viability by MTT assay and expressions of heme oxygenase-I (HO-I) and phospholylated extracellular signal-regulated protein kinase 1/2 (ERK1/2) by Western blotting.

Results: The cell viability decreased dramatically following OGD. Pretreatment with minocycline (O.I-IO JJ.mol/L) induced a significant increase in the cell viability after OGD and caused up-regulation of HO-I protein and enhanced ERK1/2 phospholylation, and the effects were especially obvious with 1 JJ.mol/L minocycline and were abolished by inhibition of ERK1/2 activity with UOI26 (IO JJ.mol/L).

Conclusion: Minocycline can protect PCI2 cells against OGD-induced toxicity by up-regulating HO-I protein expression through ERKl/2 signaling pathways.

MeSH terms

  • Animals
  • Brain Ischemia
  • Cell Hypoxia
  • Cell Survival
  • Glucose*
  • Heme Oxygenase (Decyclizing) / metabolism*
  • MAP Kinase Signaling System*
  • Minocycline / pharmacology*
  • Oxygen*
  • PC12 Cells
  • Rats
  • Up-Regulation

Substances

  • Heme Oxygenase (Decyclizing)
  • Hmox1 protein, rat
  • Minocycline
  • Glucose
  • Oxygen