Pseudomonas aeruginosa activates the quorum sensing LuxR response regulator through secretion of 2-aminoacetophenone

Chem Commun (Camb). 2015 Feb 21;51(15):3258-61. doi: 10.1039/c4cc10393a.

Abstract

In this study we identify a volatile compound produced by Pseudomonas aeruginosa, which can specifically activate the LuxR quorum-sensing response regulator of Vibrio fischeri. Comparative gas-chromatography analysis between P. aeruginosa wild type and a ΔlasR mutant strain implied that the active volatile is 2-aminoacetophenone. The use of synthetic 2-aminoacetophenone and in silico docking analyses verified the activity of the molecule and provided putative interacting residues within the binding site.

MeSH terms

  • Acetophenones / metabolism*
  • Aliivibrio fischeri / metabolism
  • Bacterial Proteins / genetics
  • Bacterial Proteins / metabolism*
  • Biosensing Techniques
  • Escherichia coli / genetics
  • Escherichia coli / metabolism
  • Pseudomonas aeruginosa / metabolism*
  • Quorum Sensing*
  • Repressor Proteins / genetics
  • Repressor Proteins / metabolism*
  • Trans-Activators / genetics
  • Trans-Activators / metabolism*

Substances

  • Acetophenones
  • Bacterial Proteins
  • Repressor Proteins
  • Trans-Activators
  • LuxR autoinducer binding proteins
  • 2-aminoacetophenone