Fibronectin-based scaffold domain proteins that bind myostatin: a patent evaluation of WO2014043344

Expert Opin Ther Pat. 2015 May;25(5):619-24. doi: 10.1517/13543776.2015.1007954. Epub 2015 Jan 29.

Abstract

Muscular dystrophies (MD) are commonly characterized by progressive loss of muscle mass and function. It is hypothesized that therapeutic blockade of the TGF-β ligand myostatin, a negative regulator of muscle mass, will stimulate muscle growth and restore muscle function. Although many anti-myostatin targets are currently being pursued in the clinical setting, the efficacies of the tested molecules have shown mixed results. The patent WO2014043344 describes a novel approach for myostatin inhibition using a modified fibronectin type III domain that could potentially be used to treat MD and other muscle-related pathologies.

Keywords: TGF-β; biological therapies; fibronectin; growth and differentiation factor-8; muscle wasting; muscular dystrophy; myostatin.

MeSH terms

  • Animals
  • Disease Progression
  • Drug Design
  • Fibronectins / metabolism*
  • Humans
  • Molecular Targeted Therapy
  • Muscular Diseases / drug therapy
  • Muscular Diseases / physiopathology
  • Muscular Dystrophies / drug therapy*
  • Muscular Dystrophies / physiopathology
  • Myostatin / antagonists & inhibitors*
  • Patents as Topic

Substances

  • Fibronectins
  • Myostatin