Significance of low level infliximab in the absence of anti-infliximab antibodies

World J Gastroenterol. 2015 Feb 14;21(6):1907-14. doi: 10.3748/wjg.v21.i6.1907.

Abstract

Aim: To evaluate the prevalence of double negative (DN) sera and the mechanisms responsible for DN status.

Methods: Sera of inflammatory bowel disease patients treated with infliximab (IFX) were tested for drug/antibodies to infliximab (ATI) trough levels and the proportion of DN results was compared between a commercially available double antigen ELISA (with labeled IFX as the detection antibody) and an anti-lambda ELISA (with anti-human lambda chain detection antibody). Repeat testing with lower than customary serum dilution (1:10) was performed. Patients with DN status were matched with IFX+/ATI- controls and were followed-up for subsequent development of non-transient ATI to investigate if DN status precedes ATI.

Results: Of 67 sera obtained at time of loss of response, only 6/67 (9%) were DN by anti-lambda ELISA compared to 27/67 (40%) with double antigen ELISA (P < 0.001, Fisher's Exact test). Of the latter 27 sera, 22% were also DN by anti-lambda ELISA, whereas 44% were actually IFX positive (IFX+ATI-), 30% were ATI positive (IFX-ATI+) and 4% were double positive (IFX+ATI+). Re-testing using a 1:10 dilution converted most DN results into IFX+ and /or ATI+ status. Patients with DN status had shorter survival free of non-transient ATI compared with matched controls (log rank test, P < 0.001). In 9/30 (30%) of these patients, non transient ATI occurred before and after the event at which the DN serum was obtained, supporting the view that a DN result may represent a particular time-point along the two curves of ATI titer rise and infliximab drug level decline.

Conclusion: DN status may result from false negative detection of IFX or ATI by double antigen ELISA, suggesting a transitional state of low-level immunogenicity, rather than non-immunological clearance.

Keywords: Biological therapy; Drug response; Immunology; Inflammatory bowel disease; Infliximab.

Publication types

  • Multicenter Study
  • Observational Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal / blood
  • Antibodies, Monoclonal / immunology*
  • Antibodies, Monoclonal / pharmacokinetics*
  • Biomarkers / blood
  • Case-Control Studies
  • Drug Monitoring
  • Enzyme-Linked Immunosorbent Assay
  • False Negative Reactions
  • Humans
  • Immunoglobulin G / blood*
  • Immunosuppressive Agents / blood
  • Immunosuppressive Agents / immunology*
  • Immunosuppressive Agents / pharmacokinetics*
  • Inflammatory Bowel Diseases / blood
  • Inflammatory Bowel Diseases / diagnosis
  • Inflammatory Bowel Diseases / drug therapy*
  • Inflammatory Bowel Diseases / immunology
  • Infliximab
  • Israel
  • Predictive Value of Tests
  • Serologic Tests
  • Time Factors
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors

Substances

  • Antibodies, Monoclonal
  • Biomarkers
  • Immunoglobulin G
  • Immunosuppressive Agents
  • Tumor Necrosis Factor-alpha
  • Infliximab