Growth differentiation factor-15 encodes a novel microRNA 3189 that functions as a potent regulator of cell death

Cell Death Differ. 2015 Oct;22(10):1641-53. doi: 10.1038/cdd.2015.9. Epub 2015 Feb 20.

Abstract

According to the latest version of miRBase, approximately 30% of microRNAs (miRNAs) are unique to primates, but the physiological function of the vast majority remains unknown. In this study, we identified miR-3189 as a novel, p53-regulated, primate-specific miRNA embedded in the intron of the p53-target gene GDF15. Antagonizing miR-3189 increased proliferation and sensitized cells to DNA damage-induced apoptosis, suggesting a tumor suppressor function for endogenous miR-3189. Identification of genome-wide miR-3189 targets revealed that miR-3189 directly inhibits the expression of a large number of genes involved in cell cycle control and cell survival. In addition, miR-3189 downregulated the expression of multiple p53 inhibitors resulting in elevated p53 levels and upregulation of several p53 targets including p21 (CDKN1A), GADD45A and the miR-3189 host gene GDF15, suggesting miR-3189 auto-regulation. Surprisingly, miR-3189 overexpression in p53-/- cells upregulated a subset of p53-targets including GDF15, GADD45A, and NOXA, but not CDKN1A. Consistent with these results, overexpression of miR-3189 potently induced apoptosis and inhibited tumorigenicity in vivo in a p53-independent manner. Collectively, our study identified miR-3189 as a novel, primate-specific miRNA whose effects are mediated by both p53-dependent and p53-independent mechanisms. miR-3189 may, therefore, represent a novel tool that can be utilized therapeutically to induce a potent proapoptotic effect even in p53-deficient tumors.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / physiology*
  • Cell Cycle Proteins
  • Cyclin-Dependent Kinase Inhibitor p21
  • Female
  • Genes, Tumor Suppressor*
  • Growth Differentiation Factor 15 / genetics*
  • HCT116 Cells
  • Humans
  • Introns*
  • Mice
  • MicroRNAs / genetics*
  • Nuclear Proteins
  • Sequence Alignment
  • Signal Transduction
  • Tumor Suppressor Protein p53

Substances

  • Cell Cycle Proteins
  • Cyclin-Dependent Kinase Inhibitor p21
  • GADD45A protein, human
  • GDF15 protein, human
  • Growth Differentiation Factor 15
  • MIRN3189 microRNA, human
  • MicroRNAs
  • Nuclear Proteins
  • TP53 protein, human
  • Tumor Suppressor Protein p53