Cardiovascular effects of detomidine, a new alpha 2-adrenoceptor agonist, in the conscious pony

J Vet Pharmacol Ther. 1989 Dec;12(4):378-88. doi: 10.1111/j.1365-2885.1989.tb00688.x.

Abstract

The cardiovascular effects of detomidine and xylazine were compared in six chronically instrumented, conscious ponies. Ponies were instrumented with a micromanometer in the left ventricular chamber, a Doppler flow probe on a coronary artery and sonomicrometer crystals in the left ventricular free wall. Heart rate, ventricular systolic pressure, stroke work, dP/dtmax, minute work and coronary blood flow were measured for 4 h following intravenous injection of detomidine at several doses or xylazine at 1.1 mg/kg. Both drugs caused a profound hypertensive response at 15 s post-injection. The magnitude of the pressure change did not increase with detomidine doses greater than 20 micrograms/kg. There was a dose-dependent effect on the duration of the hypertension. Bradycardia and A-V blockade of similar magnitude followed the hypertension at all drug doses. Both drugs caused a negative inotropic effect on the heart at all doses. Minute work, a mechanical index of myocardial O2 demand, and coronary flow decreased to a similar extent following all drug treatments. With the exception of a greater hypertensive response, detomidine at the dosages studied, produced cardiovascular effects that were very similar to those of the recommended dosage of xylazine.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adrenergic alpha-Agonists / pharmacology*
  • Animals
  • Blood Flow Velocity / drug effects
  • Blood Pressure / drug effects*
  • Heart / drug effects
  • Heart Rate / drug effects*
  • Horses / physiology*
  • Imidazoles / pharmacology*
  • Myocardium / metabolism
  • Oxygen Consumption / drug effects
  • Stroke Volume / drug effects
  • Xylazine / pharmacology

Substances

  • Adrenergic alpha-Agonists
  • Imidazoles
  • Xylazine
  • detomidine