A possible contribution of lipocalin-2 to the development of dermal fibrosis, pulmonary vascular involvement and renal dysfunction in systemic sclerosis

Br J Dermatol. 2015 Sep;173(3):681-9. doi: 10.1111/bjd.13779. Epub 2015 Jun 11.

Abstract

Background: Lipocalin-2 is an adipocytokine implicated in apoptosis, innate immunity, angiogenesis, and the development of chronic kidney disease.

Objectives: To investigate the role of lipocalin-2 in systemic sclerosis (SSc).

Materials and methods: Serum lipocalin-2 levels were determined by enzyme-linked immunosorbent assay in 50 patients with SSc and 19 healthy subjects. Lipocalin-2 expression was evaluated in the skin of patients with SSc and bleomycin (BLM)-treated mice and in Fli1-deficient endothelial cells by reverse transcriptase-real time polymerase chain reaction, immunoblotting and/or immunohistochemistry.

Results: Although serum lipocalin-2 levels were comparable between patients with SSc and healthy controls, the prevalence of scleroderma renal crisis was significantly higher in patients with SSc with elevated serum lipocalin-2 levels than in those with normal levels. Furthermore, serum lipocalin-2 levels inversely correlated with estimated glomerular filtration rate in patients with SSc with renal dysfunction. Among patients with SSc with normal renal function, serum lipocalin-2 levels positively correlated with skin score in patients with diffuse cutaneous SSc with disease duration of < 3 years and inversely correlated with estimated right ventricular systolic pressure in total patients with SSc. Importantly, in SSc lesional skin, lipocalin-2 expression was increased in dermal fibroblasts and endothelial cells. In BLM-treated mice, lipocalin-2 was highly expressed in dermal fibroblasts, but not in endothelial cells. On the other hand, the deficiency of transcription factor Fli1, which is implicated in SSc vasculopathy, induced lipocalin-2 expression in cultivated endothelial cells.

Conclusions: Lipocalin-2 may be involved in renal dysfunction and dermal fibrosis of SSc. Dysregulated matrix metalloproteinase-9/lipocalin-2-dependent angiogenesis due to Fli1 deficiency may contribute to the development of pulmonary arterial hypertension associated with SSc.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute-Phase Proteins / metabolism
  • Acute-Phase Proteins / physiology*
  • Adult
  • Aged
  • Animals
  • Apoptosis / physiology
  • Case-Control Studies
  • Female
  • Fibrosis / etiology
  • Fibrosis / pathology
  • Fibrosis / physiopathology
  • Glomerular Filtration Rate / physiology
  • Humans
  • Lipocalin-2
  • Lipocalins / metabolism
  • Lipocalins / physiology*
  • Lung Diseases / etiology*
  • Lung Diseases / physiopathology
  • Male
  • Mice
  • Middle Aged
  • Proto-Oncogene Proteins / metabolism
  • Proto-Oncogene Proteins / physiology*
  • Renal Insufficiency, Chronic / etiology*
  • Scleroderma, Systemic / etiology*
  • Scleroderma, Systemic / pathology
  • Scleroderma, Systemic / physiopathology
  • Skin / pathology*
  • Skin Diseases, Vascular / etiology
  • Skin Diseases, Vascular / physiopathology
  • Vascular Diseases / etiology*
  • Vascular Diseases / pathology
  • Vascular Diseases / physiopathology

Substances

  • Acute-Phase Proteins
  • LCN2 protein, human
  • Lipocalin-2
  • Lipocalins
  • Proto-Oncogene Proteins