The first stage and complete promoting activity of retinoic acid but not the analog RO-10-9359

Carcinogenesis. 1985 Apr;6(4):575-8. doi: 10.1093/carcin/6.4.575.

Abstract

Retinoic acid has the ability to act as either a weak first stage promoter or a weak complete promoter in the initiation-promotion protocol for skin carcinogenesis in the SENCAR mouse. The retinoid analog RO-10-9359 lacks this tumor promoting activity. Both retinoids however inhibit 12-O-tetradecanoylphorbol-13-acetate (TPA) promotion. Additional comparisons revealed that retinoic acid alone can induce dark keratinocytes, a characteristic of tumor promoters, while RO-10-9359 cannot. Retinoic acid but not RO-10-9359 can induce an immediate chemiluminescence response in human polymorphonuclear cells. Both retinoids, however, inhibit a TPA-induced response. Since the chemiluminescence response is believed to be due to oxygen free radical generation, the data suggest that the ability of retinoic acid but not RO-10-9359 to promote tumors and induce dark cells may be due to initial oxidative reactions at the cell membrane.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Etretinate / toxicity*
  • Female
  • Keratins / metabolism
  • Luminescent Measurements
  • Mice
  • Neutrophils / drug effects
  • Neutrophils / physiology
  • Ornithine Decarboxylase / metabolism
  • Skin Neoplasms / chemically induced*
  • Skin Neoplasms / enzymology
  • Skin Neoplasms / pathology
  • Tetradecanoylphorbol Acetate
  • Tretinoin / toxicity*

Substances

  • Tretinoin
  • Etretinate
  • Keratins
  • Ornithine Decarboxylase
  • Tetradecanoylphorbol Acetate