18-Hydroxylase activity in the Y1 adrenal cell line

Mol Cell Endocrinol. 1989 Sep;66(1):83-91. doi: 10.1016/0303-7207(89)90051-8.

Abstract

18-Hydroxylase activity, reported here for the first time in the mouse adrenal tumor cell line (Y1), was expressed in the metabolism of 11-deoxycorticosterone (DOC) and corticosterone (B). Detected after 24 h of incubation, it was more evident after 48 h and produced mostly 18-hydroxy-20 alpha-DHB from these exogenous substrates. However, 18-hydroxylation was quantitatively less significant than the metabolism of 20 alpha-reduction and 11 beta-hydroxylation (of DOC). The latter is also the predominant metabolism of progesterone in this cell line, during the conversion of cholesterol from the serum-supplemented culture media. The cytochrome P-450 11 beta activity of the Y1 cells is similar to that of the mouse in vivo which catalyzes the production of an 11 beta 18-dihydroxylated metabolite as the principal 18-hydroxylated steroid. It is different from that of other species, such as the rat and the bovine, both in terms of the ratio of 11 beta- to 18-hydroxylated metabolites and of the structure of these metabolites.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenal Cortex / enzymology*
  • Animals
  • Corticosterone / metabolism
  • Cytochrome P-450 CYP11B2
  • Cytochrome P-450 Enzyme System / metabolism*
  • Desoxycorticosterone / metabolism
  • Mice
  • Steroid Hydroxylases / metabolism*
  • Tumor Cells, Cultured

Substances

  • Desoxycorticosterone
  • Cytochrome P-450 Enzyme System
  • Steroid Hydroxylases
  • Cytochrome P-450 CYP11B2
  • Corticosterone