1,25-dihydroxyvitamin D-responsive element and glucocorticoid repression in the osteocalcin gene

Science. 1989 Dec 1;246(4934):1158-61. doi: 10.1126/science.2588000.

Abstract

The active hormonal form of vitamin D3, 1,25-dihydroxyvitamin D3[1,25(OH), which regulates cellular replication and function in many tissues and has a role in bone and calcium homeostasis, acts through a hormone receptor homologous with other steroid and thyroid hormone receptors. A 1,25(OH)2D3-responsive element (VDRE), which is within the promoter for osteocalcin [a bone protein induced by 1,25(OH)2D3] is unresponsive to other steroid hormones, can function in a heterologous promoter, and contains a doubly palindromic DNA sequence (TTGGTGACTCACCGGGTGAAC; -513 to -493 bp), with nucleotide sequence homology to other hormone responsive elements. The potent glucocorticoid repression of 1,25(OH)2D3 induction and of basal activity of this promoter acts through a region between -196 and +34 bp, distinct from the VDRE.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Calcitriol / pharmacology*
  • Chloramphenicol O-Acetyltransferase / genetics
  • DNA / genetics*
  • Dexamethasone / pharmacology
  • Gene Expression / drug effects*
  • Glucocorticoids / pharmacology*
  • Humans
  • Molecular Sequence Data
  • Osteocalcin / genetics*
  • Promoter Regions, Genetic / genetics*
  • Rats
  • Restriction Mapping
  • Sequence Homology, Nucleic Acid
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Glucocorticoids
  • Osteocalcin
  • Dexamethasone
  • DNA
  • Chloramphenicol O-Acetyltransferase
  • Calcitriol