Moxidectin steady state prior to inoculation protects cats from subsequent, repeated infection with Dirofilaria immitis

Parasit Vectors. 2015 Feb 18:8:107. doi: 10.1186/s13071-015-0710-z.

Abstract

Background: Infection of cats with Dirofilaria immitis causes seroconversion on antibody tests and pulmonary pathology, often without subsequent development of adult heartworms. Consistent administration of topical 10% imidacloprid-1% moxidectin has been shown to result in sustained plasma levels of moxidectin in cats after three to five treatments, a pharmacokinetic behavior known as "steady state".

Methods: To evaluate the ability of moxidectin at "steady state" to protect cats from subsequent infection with D. immitis, cats (n = 10) were treated with the labeled dose of topical 10% imidacloprid-1% moxidectin for four monthly treatments. Each cat was inoculated with 25 third-stage larvae of D. immitis 7, 14, 21, and 28 days after the last treatment; non-treated cats (n = 9) were inoculated on the same days, serving as infection controls. Blood samples were collected from each cat from 1 month prior to treatment until 7 months after the final inoculation and tested for antibody to, and antigen and microfilaria of, D. immitis.

Results: Measurement of serum levels of moxidectin confirmed steady state in treated cats. Cats treated with topical 10% imidacloprid-1% moxidectin prior to trickle inoculation of D. immitis L3 larvae throughout the 28 day post-treatment period remained negative on antibody and antigen tests throughout the study and did not develop gross or histologic lesions characteristic of heartworm infection. A majority of non-treated cats tested antibody positive by 3-4 months post infection (6/9) and, after heat treatment, tested antigen positive by 6-7 months post-infection (5/9). Histologic lesions characteristic of D. immitis infection, including intimal and medial thickening of the pulmonary artery, were present in every cat with D. immitis antibodies (6/6), although adult D. immitis were confirmed in only 5/6 antibody-positive cats at necropsy. Microfilariae were not detected at any time.

Conclusions: Taken together, these data indicate that prior treatment with 10% imidacloprid-1% moxidectin protected cats from subsequent infection with D. immitis for 28 days, preventing both formation of a detectable antibody response and development of pulmonary lesions by either immature stages of D. immitis or young adult heartworms.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Topical
  • Animals
  • Anthelmintics / administration & dosage*
  • Anthelmintics / pharmacokinetics
  • Antibodies, Helminth / blood
  • Antigens, Helminth / blood
  • Cat Diseases / parasitology
  • Cat Diseases / prevention & control*
  • Cats
  • Chemoprevention / methods*
  • Dirofilaria immitis / isolation & purification*
  • Dirofilariasis / parasitology
  • Dirofilariasis / prevention & control*
  • Macrolides / administration & dosage*
  • Macrolides / pharmacokinetics
  • Plasma / chemistry
  • Treatment Outcome

Substances

  • Anthelmintics
  • Antibodies, Helminth
  • Antigens, Helminth
  • Macrolides
  • moxidectin