IκBβ enhances the generation of the low-affinity NFκB/RelA homodimer

Nat Commun. 2015 May 7:6:7068. doi: 10.1038/ncomms8068.

Abstract

The NFκB family of dimeric transcription factors regulate inflammatory and immune responses. While the dynamic control of NFκB dimer activity via the IκB-NFκB signalling module is well understood, there is little information on how specific dimer repertoires are generated from Rel family polypeptides. Here we report the iterative construction-guided by in vitro and in vivo experimentation-of a mathematical model of the Rel-NFκB generation module. Our study reveals that IκBβ has essential functions within the Rel-NFκB generation module, specifically for the RelA:RelA homodimer, which controls a subset of NFκB target genes. Our findings revise the current dogma of the three classical, functionally related IκB proteins by distinguishing between a positive 'licensing' factor (IκBβ) that contributes to determining the available NFκB dimer repertoire in a cell's steady state, and negative feedback regulators (IκBα and -ɛ) that determine the duration and dynamics of the cellular response to an inflammatory stimulus.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Binding, Competitive
  • Biophysical Phenomena
  • I-kappa B Proteins / metabolism*
  • Kinetics
  • Mice
  • Models, Biological
  • NF-kappa B / metabolism*
  • Protein Binding
  • Protein Isoforms / metabolism
  • Protein Multimerization*
  • Signal Transduction
  • Transcription Factor RelA / metabolism*

Substances

  • I kappa B beta protein
  • I-kappa B Proteins
  • NF-kappa B
  • Protein Isoforms
  • Transcription Factor RelA