Development of a highly thermostable, adjuvanted human papillomavirus vaccine

Eur J Pharm Biopharm. 2015 Aug:94:220-8. doi: 10.1016/j.ejpb.2015.05.009. Epub 2015 May 18.

Abstract

A major impediment to economical, worldwide vaccine distribution is the requirement for a "cold chain" to preserve antigenicity. We addressed this problem using a model human papillomavirus (HPV) vaccine stabilized by immobilizing HPV16 L1 capsomeres, i.e., pentameric subunits of the virus capsid, within organic glasses formed by lyophilization. Lyophilized glass and liquid vaccine formulations were incubated at 50°C for 12weeks, and then analyzed for retention of capsomere conformational integrity and the ability to elicit neutralizing antibody responses after immunization of BALB/c mice. Capsomeres in glassy-state vaccines retained tertiary and quaternary structure, and critical conformational epitopes. Moreover, glassy formulations adjuvanted with aluminum hydroxide or aluminum hydroxide and glycopyranoside lipid A were not only as immunogenic as the commercially available HPV vaccine Cervarix®, but also retained complete neutralizing immunogenicity after high-temperature storage. The thermal stability of such adjuvanted vaccine powder preparations may thus eliminate the need for the cold chain.

Keywords: Aluminum hydroxide; Glycopyranoside lipid A; Human papillomavirus; Lyophilization; Stability; Vaccine.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adjuvants, Immunologic / chemistry*
  • Animals
  • Antibodies, Neutralizing / blood
  • Antibodies, Viral / blood
  • Calorimetry, Differential Scanning
  • Capsid Proteins / biosynthesis
  • Capsid Proteins / genetics
  • Capsid Proteins / immunology*
  • Dose-Response Relationship, Drug
  • Drug Stability
  • Drug Storage
  • Electrophoresis, Polyacrylamide Gel
  • Enzyme-Linked Immunosorbent Assay
  • Epitopes / chemistry
  • Female
  • Freeze Drying
  • Mice, Inbred BALB C
  • Microscopy, Electron, Transmission
  • Neutralization Tests
  • Oncogene Proteins, Viral / genetics
  • Oncogene Proteins, Viral / immunology*
  • Papillomavirus Vaccines / chemistry*
  • Papillomavirus Vaccines / immunology*
  • Protein Conformation
  • Spectrometry, Fluorescence
  • Temperature

Substances

  • Adjuvants, Immunologic
  • Antibodies, Neutralizing
  • Antibodies, Viral
  • Capsid Proteins
  • Epitopes
  • HPV L1 protein, Human papillomavirus
  • Oncogene Proteins, Viral
  • Papillomavirus Vaccines
  • human papillomavirus vaccine, L1 type 16, 18