Cripto-1 as a novel therapeutic target for triple negative breast cancer

Oncotarget. 2015 May 20;6(14):11910-29. doi: 10.18632/oncotarget.4182.

Abstract

Triple-negative breast cancer (TNBC) presents the poorest prognosis among the breast cancer subtypes and no current standard therapy. Here, we performed an in-depth molecular analysis of a mouse model that establishes spontaneous lung metastasis from JygMC(A) cells. These primary tumors resembled the triple-negative breast cancer (TNBC) both phenotypically and molecularly. Morphologically, primary tumors presented both epithelial and spindle-like cells but displayed only adenocarcinoma-like features in lung parenchyma. The use of laser-capture microdissection combined with Nanostring mRNA and microRNA analysis revealed overexpression of either epithelial and miRNA-200 family or mesenchymal markers in adenocarcinoma and mesenchymal regions, respectively. Cripto-1, an embryonic stem cell marker, was present in spindle-like areas and its promoter showed activity in primary tumors. Cripto-1 knockout by the CRISPR-Cas9 system inhibited tumor growth and pulmonary metastasis. Our findings show characterization of a novel mouse model that mimics the TNBC and reveal Cripto-1 as a TNBC target hence may offer alternative treatment strategies for TNBC.

Trial registration: ClinicalTrials.gov NCT01151449.

Keywords: Cripto-1; Notch4; epithelial-mesenchymal plasticity; mouse model; triple-negative breast cancer.

Publication types

  • Research Support, N.I.H., Intramural

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Cell Transformation, Neoplastic / metabolism*
  • Epidermal Growth Factor / metabolism*
  • Epithelial-Mesenchymal Transition / physiology
  • Female
  • Fluorescent Antibody Technique
  • Gene Knockout Techniques
  • Immunohistochemistry
  • In Situ Nick-End Labeling
  • Laser Capture Microdissection
  • Mammary Neoplasms, Experimental / metabolism
  • Mammary Neoplasms, Experimental / pathology*
  • Membrane Glycoproteins / metabolism*
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Neoplasm Proteins / metabolism*
  • Oligonucleotide Array Sequence Analysis
  • Polymerase Chain Reaction
  • Triple Negative Breast Neoplasms / metabolism
  • Triple Negative Breast Neoplasms / pathology*

Substances

  • Membrane Glycoproteins
  • Neoplasm Proteins
  • Tdgf1 protein, mouse
  • Epidermal Growth Factor

Associated data

  • ClinicalTrials.gov/NCT01151449