Concomitant immune-related events in Wilson disease: implications for monitoring chelator therapy

J Inherit Metab Dis. 2016 Jan;39(1):125-30. doi: 10.1007/s10545-015-9866-0. Epub 2015 Jun 12.

Abstract

Background and aims: Current guidelines favor the use of chelating agents (d-penicillamine, trientine) in first line therapy of symptomatic Wilson disease patients. Development of chelator induced immunological adverse events are a concern especially under d-penicillamine therapy. This study assessed the prevalence of co-existing or therapy-related immune-mediated diseases in Wilson disease patients, and evaluated the role of antinuclear antibodies in therapy monitoring.

Methods: We retrospectively analyzed 235 Wilson disease patients. Medical regimens were classified and analyzed in relation to adverse events and antinuclear antibody courses.

Results: Coexisting immune-mediated diseases were evident in 19/235 (8.1%) patients, of which 13/235 (5.5%) had pre-existing autoimmune diseases. Six patients (2.6%) developed an autoimmune disease under therapy, all of them under long-term d-penicillamine treatment. Data relating to antinuclear antibody courses during treatment and adverse events were available for patients treated with d-penicillamine (n = 91), trientine (n = 58), and zinc salts (n = 58). No significant increase in antinuclear antibody titers in patients treated with d-penicillamine (16/91; 17.6%), trientine (12/58; 20.7%), and zinc (7/58; 12.1%) were found.

Conclusion: Under long-term d-penicillamine therapy a minority of patients developed immune-mediated disease. Elevations in antinuclear antibodies were found frequently, but no correlations were evident between increases in antinuclear antibodies and the development of immune-mediated diseases or medical regimes. Thus, the value of antinuclear antibodies for monitoring adverse events under chelator therapy seems to be limited.

MeSH terms

  • Adolescent
  • Adult
  • Antibodies, Antinuclear / immunology
  • Autoimmune Diseases / chemically induced
  • Autoimmune Diseases / immunology
  • Chelating Agents / adverse effects*
  • Chelating Agents / therapeutic use*
  • Child
  • Cross-Sectional Studies
  • Drug Monitoring / methods
  • Drug-Related Side Effects and Adverse Reactions / immunology*
  • Female
  • Hepatolenticular Degeneration / drug therapy*
  • Hepatolenticular Degeneration / immunology*
  • Humans
  • Male
  • Penicillamine / adverse effects
  • Penicillamine / immunology
  • Penicillamine / therapeutic use
  • Retrospective Studies
  • Trientine / adverse effects
  • Trientine / immunology
  • Trientine / therapeutic use
  • Young Adult
  • Zinc / adverse effects
  • Zinc / immunology
  • Zinc / therapeutic use

Substances

  • Antibodies, Antinuclear
  • Chelating Agents
  • Penicillamine
  • Zinc
  • Trientine