A new 3-alkylpyridine alkaloid from the marine sponge Haliclona sp. and its cytotoxic activity

Nat Prod Res. 2016 Jun;30(11):1262-5. doi: 10.1080/14786419.2015.1054826. Epub 2015 Jul 13.

Abstract

A new alkaloid, 3-dodecyl pyridine containing a terminal cyano group (1), was isolated from the methanol extract of an Indonesia marine sponge Haliclona sp. Its chemical structure was determined by a combination of spectroscopic methods, including 1D and 2D NMR. Bioassay results indicated that compound 1 had moderate cytotoxity against tumour cell lines A549, MCF-7 and Hela with IC50 values of 41.8, 48.4 and 33.2 μM, respectively.

Keywords: 3-alkylpyridine; Haliclona sp.; alkaloid; cytotoxicity.

MeSH terms

  • Alkaloids / chemistry*
  • Alkaloids / toxicity
  • Animals
  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / isolation & purification*
  • Antineoplastic Agents / pharmacology
  • Cell Line, Tumor
  • Haliclona / chemistry*
  • Humans
  • Indonesia
  • Inhibitory Concentration 50
  • Magnetic Resonance Spectroscopy
  • Molecular Structure
  • Porifera / chemistry
  • Pyridines / isolation & purification

Substances

  • Alkaloids
  • Antineoplastic Agents
  • Pyridines
  • pyridine