Suitability of long-acting metoclopramide for prophylaxis of chemotherapy-induced delayed nausea and vomiting

Arzneimittelforschung. 1989 Nov;39(11):1464-7.

Abstract

Delayed nausea and emesis are common after cancer chemotherapy, especially cisplatin-containing regimens. Often no, or inadequate, prophylactic antiemetic cover is prescribed in these usually ambulant patients. Metoclopramide is a very effective drug in preventing the acute emetic and nauseating effects of cisplatin. The long-acting metoclopramide formulations (in the present study: Gastrosil retard) may be effective in preventing the delayed toxicity. 12-hourly dosing of 60 mg long-acting metoclopramide in a typical oncology ward situation led to stable metoclopramide levels of approximately 100ng/ml in the observed 74 h in 18 patients, with the well-known wide plasma concentration variability. The clinical efficacy of long-acting metoclopramide in this indication remains to be evaluated.

MeSH terms

  • Antineoplastic Agents / adverse effects*
  • Antineoplastic Agents / therapeutic use
  • Chromatography, High Pressure Liquid
  • Humans
  • Metoclopramide / administration & dosage
  • Metoclopramide / pharmacokinetics
  • Metoclopramide / therapeutic use*
  • Nausea / chemically induced
  • Nausea / drug therapy*
  • Neoplasms / drug therapy
  • Vomiting / chemically induced
  • Vomiting / drug therapy*

Substances

  • Antineoplastic Agents
  • Metoclopramide