Pharmacokinetics of atracurium besylate in the pig after a single i.v. injection

Eur J Drug Metab Pharmacokinet. 1989 Oct-Dec;14(4):299-302. doi: 10.1007/BF03190115.

Abstract

A pharmacokinetic study of atracurium besylate was performed in the pig after a single i.v. bolus injection of 2 mg/kg, the dose needed to produce surgical neuromuscular blockade. The plasma concentration values were obtained by high performance liquid chromatography. Using a two-compartment pharmacokinetic model, the elimination half life was found to be 28.6 +/- 6.3 min (mean +/- SEM), the total volume of distribution 341 +/- 56 ml/kg and the plasma clearance 8.7 +/- 1.1 ml/min/kg. Although the doses required to obtain a satisfactory neuromuscular blockade as well as the plasma level, volume of distribution and plasma clearance values were higher in the pig than in man, the distribution and elimination half-lives were similar to those recently reported.

MeSH terms

  • Animals
  • Atracurium / administration & dosage
  • Atracurium / pharmacokinetics*
  • Chromatography, High Pressure Liquid
  • Half-Life
  • Injections, Intravenous
  • Swine

Substances

  • Atracurium