Total Synthesis of Lignan Lactone (-)-Hinokinin

Nat Prod Bioprospect. 2015 Oct;5(5):255-61. doi: 10.1007/s13659-015-0073-3. Epub 2015 Oct 12.

Abstract

This research paper is aimed at studying the total synthesis of pharmacologically active lignan (-)-hinokinin. The synthesis features a three-step cascade reaction involving highly stereoselective Michael addition, anion-oxidative hydroxylation, and oxygen anion cyclization to construct the pivotal butyrolactonimidate intermediate.

Keywords: Cascade reaction; Hinokinin; Lignan; Total synthesis.