Cyclosporin A: action and side-effects

Toxicol Lett. 1989 Mar;46(1-3):125-39. doi: 10.1016/0378-4274(89)90122-7.

Abstract

Cyclosporin A (CSA) is a new, potent immunosuppressive agent which is of proven value in organ transplantation. The use of CSA is associated with numerous side-effects, of which a dose-dependent nephrotoxicity is the most serious. CSA nephrotoxicity can be divided into two major groups: (i) functional toxicity without significant morphological lesions and (ii) morphological forms of toxicity with tubular and/or vascular-interstitial lesions. Vascular-interstitial toxicity is the most serious form because the renal lesions are irreversible.

Publication types

  • Review

MeSH terms

  • Acute Kidney Injury / chemically induced*
  • Acute Kidney Injury / pathology
  • Cyclosporins / adverse effects*
  • Cyclosporins / pharmacokinetics
  • Cyclosporins / therapeutic use
  • Humans
  • Kidney Tubular Necrosis, Acute / chemically induced
  • Nephritis, Interstitial / chemically induced*
  • Nephritis, Interstitial / pathology

Substances

  • Cyclosporins