Ticagrelor vs. clopidogrel in non-ST-elevation acute coronary syndromes

Herz. 2016 May;41(3):246-9. doi: 10.1007/s00059-015-4359-3. Epub 2015 Nov 2.

Abstract

Aim: The aim of this study was to evaluate the bradyarrhythmic events associated with ticagrelor combination therapy in the management of patients presenting with non-ST-segment elevation myocardial infarction (NSTEMI).

Patients and methods: The study comprised 300 patients with NSTEMI who were treated via percutaneous coronary intervention (PCI). Patients were randomly assigned to two groups: the clopidogrel group (initial dose of 300 mg and then maintenance dose of 75 mg once daily, n = 151) and the ticagrelor group (initial dose of 180 mg and then maintenance dose of 90 mg twice daily, n = 149). All patients were followed up in the outpatient clinic. Follow-up included 12-lead electrocardiography and 24-h Holter monitoring performed 1, 6, and 12 months after the revascularization procedure.

Results: Of the 300 patients, 112 patients (36.7 %) had a decrease in heart rate at the 12-month follow-up. Of these, 80 patients were in the ticagrelor group (53.3 %) vs. 32 patients in the clopidogrel group (24.7 %; p < 0.05). However, the difference was not statistically significant at the 1-month and 6-month follow-up visits. After adjusting for potential confounders, the reduction in heart rate with ticagrelor combination therapy remained independently associated with a reduced risk of major adverse cardiovascular events (hazard ratio, 2.1; 95 % CI, 1.90-2.23), while ticagrelor therapy reduced the risk to a level equivalent to that of patients in the clopidogrel group.

Conclusion: Ticagrelor can lower the resting heart rate of patients and cause bradyarrhythmias in the 12th month after PCI.

Keywords: Bradyarrhythmia; Clopidogrel; Coronary artery disease; Non-ST-segment MI; Ticagrelor.

MeSH terms

  • Acute Coronary Syndrome / drug therapy*
  • Acute Coronary Syndrome / mortality*
  • Adenosine / administration & dosage
  • Adenosine / adverse effects
  • Adenosine / analogs & derivatives*
  • Bradycardia / chemically induced
  • Bradycardia / mortality
  • Clopidogrel
  • Comorbidity
  • Electrocardiography / drug effects
  • Female
  • Germany / epidemiology
  • Humans
  • Male
  • Non-ST Elevated Myocardial Infarction / drug therapy*
  • Non-ST Elevated Myocardial Infarction / mortality*
  • Prevalence
  • Purinergic P2Y Receptor Antagonists / administration & dosage
  • Risk Factors
  • Survival Rate
  • Ticagrelor
  • Ticlopidine / administration & dosage
  • Ticlopidine / analogs & derivatives*
  • Treatment Outcome

Substances

  • Purinergic P2Y Receptor Antagonists
  • Clopidogrel
  • Ticagrelor
  • Adenosine
  • Ticlopidine