Cytotoxic Activities of Eosinophil Cationic Protein and Eosinophil-derived Neurotoxin: In Silico Analysis

Cancer Genomics Proteomics. 2015 Nov-Dec;12(6):397-402.

Abstract

Background: Eosinophil cationic protein (ECP) and eosinophil derived-neurotoxin (EDN) are homologous ribonuclease (RNAse) A family proteins. The objective of the present study was to in silico characterize ECP and EDN with respect to their cytotoxic activities.

Materials and methods: Structural, physicochemical, and conserved domain characterizations were carried-out using open-source software, such as InterProScan, NetOGlyc, NetPhos and Discovery Studio 3.1.

Results: The proteins did not have atypical conserved domains. EDN had a greater number of glutamine amino acid residues, whereas ECP had a predominance of arginine. ECP had four possible N-glycosylation, three O-glycosylation and four phosphorylation sites. EDN had five putative N-glycosylation, three phosphorylation and no O-glycosylation sites.

Conclusion: The greater cationicity of ECP may be related to its higher cytotoxicity and to the fact that the varying post-translational modification profiles can generate functional differences from structural alteration. In vivo and in vitro studies need to be performed in order to confirm these predictions.

Keywords: Eosinophil cationic protein; bioinformatics; eosinophil-derived neurotoxin; homology; post-translational modifications.

MeSH terms

  • Arginine / chemistry
  • Computational Biology
  • Databases, Protein
  • Eosinophil Cationic Protein / metabolism*
  • Eosinophil-Derived Neurotoxin / metabolism*
  • Gene Expression Regulation*
  • Glutamine / chemistry
  • Glycosylation
  • Humans
  • Protein Processing, Post-Translational
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Ribonuclease, Pancreatic / chemistry
  • Software

Substances

  • Glutamine
  • Arginine
  • Eosinophil-Derived Neurotoxin
  • Eosinophil Cationic Protein
  • Ribonuclease, Pancreatic