DBU-mediated metal-free oxidative cyanation of α-amino carbonyl compounds: using molecular oxygen as the oxidant

Org Biomol Chem. 2016 Jan 7;14(1):165-71. doi: 10.1039/c5ob01690h. Epub 2015 Nov 18.

Abstract

A novel DBU-mediated oxidative cyanation of α-amino carbonyl compounds by using air as the sole oxidant was developed under mild metal-free conditions for the first time. The reaction involves a tandem oxidation/Strecker reaction/oxidation process and provides a new and efficient method for the construction of α-iminonitriles in good to high yields in a single step.

Publication types

  • Research Support, Non-U.S. Gov't