Amino acid-dependent NPRL2 interaction with Raptor determines mTOR Complex 1 activation

Cell Signal. 2016 Feb;28(2):32-41. doi: 10.1016/j.cellsig.2015.11.008. Epub 2015 Nov 12.

Abstract

We assign a new function to a tumor suppressor NPRL2 that activates the mTOR complex 1 (mTORC1) activity. The positive regulation of mTORC1 activity by NPRL2 is mediated through NPRL2 interaction with Raptor. While NPRL2 interacts with Rag GTPases, RagD in particular, to interfere with mTORC1 activity in amino acid scarcity, NPRL2 interacts with Raptor in amino acid sufficiency to activate mTORC1. A reciprocal relationship exists between NPRL2 binding to Rag GTPases and Raptor. NPRL2 majorly locates in the lysosomal membranes and has a higher binding affinity to the dominant negative mutant heterodimer of RagA(GDP)/RagD(GTP) that inactivates mTORC1. However, the binding affinity of NPRL2 with Raptor is much less pronounced in cells expressing the dominant negative mutant heterodimer of RagA(GDP)/RagD(GTP) than in cells expressing the dominant positive mutant heterodimer, RagA(GTP)/RagD(GDP). The positive effect of NPRL2 on TORC1 pathway was also evidenced in Drosophila animal model. Here, we propose a 'seesaw' model in which the interactive behavior of NPRL2 with Raptor determines mTORC1 activation by amino acid signaling in animal cells.

Keywords: Amino acids; Lysosome; NPRL2; Rag GTPases; Raptor; mTOR complex 1 (mTORC1).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing / metabolism*
  • Amino Acids / metabolism*
  • GTPase-Activating Proteins / metabolism
  • HEK293 Cells
  • Humans
  • Mechanistic Target of Rapamycin Complex 1
  • Models, Biological
  • Monomeric GTP-Binding Proteins / metabolism
  • Multiprotein Complexes / metabolism*
  • Protein Binding
  • Regulatory-Associated Protein of mTOR
  • Signal Transduction
  • TOR Serine-Threonine Kinases / metabolism*
  • Tumor Suppressor Proteins / metabolism*

Substances

  • Adaptor Proteins, Signal Transducing
  • Amino Acids
  • GTPase-Activating Proteins
  • Multiprotein Complexes
  • NPRL2 protein, human
  • NPRL3 protein, human
  • RPTOR protein, human
  • Regulatory-Associated Protein of mTOR
  • Tumor Suppressor Proteins
  • Mechanistic Target of Rapamycin Complex 1
  • TOR Serine-Threonine Kinases
  • Monomeric GTP-Binding Proteins