Oral ixazomib maintenance therapy in multiple myeloma

Expert Rev Anticancer Ther. 2016;16(1):21-32. doi: 10.1586/14737140.2016.1123627.

Abstract

Continuous therapy has proven to be an effective therapeutic strategy to improve the outcome of both young and elderly multiple myeloma patients. Remarkably, lenalidomide and bortezomib showed to play a crucial role in this setting due to their safety profile allowing long-term exposure. Ixazomib, the first oral proteasome inhibitor to be evaluated in multiple myeloma, exerts substantial anti-myeloma activity as a single agent and particularly in combination with immunomodulatory drugs and it may be an attractive option for maintenance therapy. Here we address the issue of maintenance therapy as part of a therapeutic approach of multiple myeloma patients focusing on the potential role of ixazomib.

Keywords: Ixazomib; maintenance; minimal residual disease; multiple myeloma; proteasome inhibitors.

Publication types

  • Review

MeSH terms

  • Administration, Oral
  • Antineoplastic Agents / administration & dosage*
  • Antineoplastic Agents / adverse effects
  • Antineoplastic Agents / pharmacology
  • Boron Compounds / administration & dosage*
  • Boron Compounds / adverse effects
  • Boron Compounds / pharmacology
  • Glycine / administration & dosage
  • Glycine / adverse effects
  • Glycine / analogs & derivatives*
  • Glycine / pharmacology
  • Humans
  • Multiple Myeloma / drug therapy*
  • Multiple Myeloma / pathology
  • Proteasome Inhibitors / administration & dosage
  • Proteasome Inhibitors / adverse effects
  • Proteasome Inhibitors / pharmacology

Substances

  • Antineoplastic Agents
  • Boron Compounds
  • Proteasome Inhibitors
  • ixazomib
  • Glycine