Chiral Boron Complex-Promoted Asymmetric Diels-Alder Cycloaddition and Its Application in Natural Product Synthesis

J Org Chem. 2016 Jan 15;81(2):458-68. doi: 10.1021/acs.joc.5b02248. Epub 2015 Dec 22.

Abstract

An efficient method for the asymmetric Diels-Alder cycloaddition of 2'-hydroxychalcones with acyclic or cyclic dienes has been successfully developed. The Diels-Alder cycloaddition is mediated by a chiral boron complex with VANOL, affording the corresponding products in high yields and with excellent diastereo- and enantioselectivities. This reaction enabled the enantioselective construction of cyclohexene skeletons crucial for the total synthesis of a number of Diels-Alder-type natural products (-)-nicolaioidesin C, (-)-panduratine A, (-)-kuwanon I, (+)-kuwanon J, and (-)-brosimones A and B.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biological Products / chemical synthesis*
  • Biological Products / chemistry
  • Boron Compounds / chemistry*
  • Chalcones / chemistry*
  • Cycloaddition Reaction
  • Cyclohexenes / chemistry*
  • Stereoisomerism

Substances

  • Biological Products
  • Boron Compounds
  • Chalcones
  • Cyclohexenes
  • cyclohexene
  • 2'-hydroxychalcone