Contractile effect of endothelin on isolated iris sphincter muscle of the pig

Eur J Pharmacol. 1989 Sep 1;168(1):119-21. doi: 10.1016/0014-2999(89)90643-2.

Abstract

Porcine endothelin (1 nM-0.3 microM) produced a concentration-dependent contraction of the isolated sphincter muscle of the pig iris. Neither atropine (1 microM) nor tetrodotoxin (1 microM) nor pre-exposure of the preparation to 10 microM capsaicin for 15 min affected the endothelin-induced response. We propose that the endothelin-induced contraction of the iris sphincter muscle of the pig is largely due to a direct action on smooth muscle cells and is unrelated to neurogenic myotic mechanisms.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Atropine / pharmacology
  • Capsaicin / pharmacology
  • Endothelins
  • In Vitro Techniques
  • Iris / drug effects
  • Muscle Contraction / drug effects
  • Muscle, Smooth / drug effects*
  • Peptides / pharmacology*
  • Swine
  • Tetrodotoxin / pharmacology

Substances

  • Endothelins
  • Peptides
  • Tetrodotoxin
  • Atropine
  • Capsaicin