Treatment with abatacept prevents experimental dermal fibrosis and induces regression of established inflammation-driven fibrosis

Ann Rheum Dis. 2016 Dec;75(12):2142-2149. doi: 10.1136/annrheumdis-2015-208213. Epub 2016 Feb 24.

Abstract

Objective: Activated T cells are the main component of the inflammatory skin infiltrates that characterise systemic sclerosis (SSc). Our aim was to investigate the efficacy of abatacept, which tempers T-cell activation, in reducing skin fibrosis in complementary mouse models of SSc.

Methods: The antifibrotic properties of abatacept were evaluated in the mouse models of bleomycin-induced dermal fibrosis and sclerodermatous chronic graft-versus-host disease, reflecting early and inflammatory stages of SSc. Thereafter, we studied the efficacy of abatacept in tight skin (Tsk-1) mice, an inflammation-independent mouse model of skin fibrosis.

Results: Abatacept efficiently prevented bleomycin-induced skin fibrosis and was also effective in the treatment of established fibrosis. In this model, abatacept decreased total and activated T-cell, B-cell and monocyte infiltration in the lesional skin. Abatacept did not protect CB17-SCID mice from the development of bleomycin-induced dermal fibrosis, which supports that T cells are necessary to drive the antifibrotic effects of abatacept. Upon bleomycin injections, skin interleukin (IL) 6 and IL-10 levels were significantly reduced upon abatacept treatment. Moreover, treatment with abatacept ameliorated fibrosis in the chronic graft-versus-host disease model, but demonstrated no efficacy in Tsk-1 mice. The tolerance of abatacept was excellent in the three mouse models.

Conclusions: Using complementary models, we demonstrate that inhibition of T-cell activation by abatacept can prevent and induce the regression of inflammation-driven dermal fibrosis. Translation to human disease is now required, and targeting early and inflammatory stages of SSc sounds the most appropriate for positioning abatacept in SSc.

Keywords: Inflammation; Systemic Sclerosis; T Cells.

MeSH terms

  • Abatacept / pharmacology*
  • Animals
  • B-Lymphocytes / drug effects
  • Bleomycin
  • Disease Models, Animal
  • Fibrosis
  • Graft vs Host Disease / drug therapy
  • Interleukin-10 / metabolism
  • Interleukin-6 / metabolism
  • Lymphocyte Activation / drug effects*
  • Mice
  • Scleroderma, Systemic / chemically induced
  • Scleroderma, Systemic / drug therapy*
  • Scleroderma, Systemic / pathology*
  • Skin Diseases / chemically induced
  • Skin Diseases / pathology*
  • Skin Diseases / prevention & control*
  • T-Lymphocytes / drug effects*

Substances

  • IL10 protein, mouse
  • Interleukin-6
  • interleukin-6, mouse
  • Bleomycin
  • Interleukin-10
  • Abatacept