A Chimeric Switch-Receptor Targeting PD1 Augments the Efficacy of Second-Generation CAR T Cells in Advanced Solid Tumors

Cancer Res. 2016 Mar 15;76(6):1578-90. doi: 10.1158/0008-5472.CAN-15-2524.

Abstract

Chimeric antigen receptor (CAR)-modified adoptive T-cell therapy has been successfully applied to the treatment of hematologic malignancies, but faces many challenges in solid tumors. One major obstacle is the immune-suppressive effects induced in both naturally occurring and genetically modified tumor-infiltrating lymphocytes (TIL) by inhibitory receptors (IR), namely PD1. We hypothesized that interfering with PD1 signaling would augment CAR T-cell activity against solid tumors. To address this possibility, we introduced a genetically engineered switch receptor construct, comprising the truncated extracellular domain of PD1 and the transmembrane and cytoplasmic signaling domains of CD28, into CAR T cells. We tested the effect of this supplement, "PD1CD28," on human CAR T cells targeting aggressive models of human solid tumors expressing relevant tumor antigens. Treatment of mice bearing large, established solid tumors with PD1CD28 CAR T cells led to significant regression in tumor volume due to enhanced CAR TIL infiltrate, decreased susceptibility to tumor-induced hypofunction, and attenuation of IR expression compared with treatments with CAR T cells alone or PD1 antibodies. Taken together, our findings suggest that the application of PD1CD28 to boost CAR T-cell activity is efficacious against solid tumors via a variety of mechanisms, prompting clinical investigation of this potentially promising treatment modality.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Antigens, Neoplasm / immunology
  • CD28 Antigens / immunology
  • Cell Line, Tumor
  • Female
  • Humans
  • Immunotherapy, Adoptive / methods
  • K562 Cells
  • Lymphocytes, Tumor-Infiltrating / immunology
  • Mice
  • Mice, Inbred NOD
  • Mice, SCID
  • Neoplasms / immunology*
  • Programmed Cell Death 1 Receptor / immunology*
  • Receptors, Antigen, T-Cell / immunology
  • Signal Transduction / immunology
  • T-Lymphocytes / immunology*
  • Tumor Burden / immunology
  • Xenograft Model Antitumor Assays / methods

Substances

  • Antigens, Neoplasm
  • CD28 Antigens
  • Programmed Cell Death 1 Receptor
  • Receptors, Antigen, T-Cell