Hypoxia-responsive miR-124 and miR-144 reduce hypoxia-induced autophagy and enhance radiosensitivity of prostate cancer cells via suppressing PIM1

Cancer Med. 2016 Jun;5(6):1174-82. doi: 10.1002/cam4.664. Epub 2016 Mar 14.

Abstract

Cancer cells in hypoxia usually make adaptive changes in cellular metabolism, such as altered autophagy. This might be a cause of enhanced radioresistance in some types of cancer. In this study, we investigated hypoxia-responsive miRNAs in two prostate cancer cell lines (DU145 and PC3). This study firstly reported that hypoxia induces further downregulation of miR-124 and miR-144, which might be a result of impaired dicer expression. These two miRNAs can simultaneously target 3'UTR of PIM1. Functional study showed that miR-124 or miR-144 overexpression can inhibit hypoxia-induced autophagy and enhance radiosensitivity at least via downregulating PIM1. Therefore, hypoxia induced miR-124 and miR-144 downregulation may contribute to a prosurvival mechanism of prostate cancer cells to hypoxia and irradiation at least through attenuated suppressing of PIM1. This finding presents a potential therapeutic target for prostate cancer.

Keywords: Autophagy; PIM1; hypoxia; miR-124; miR-144; radiosensitivity.

MeSH terms

  • 3' Untranslated Regions
  • Autophagy / genetics*
  • Base Sequence
  • Binding Sites
  • Cell Line, Tumor
  • Cluster Analysis
  • Down-Regulation
  • Gene Expression Profiling
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Hypoxia / genetics*
  • Hypoxia / metabolism
  • Male
  • MicroRNAs / chemistry
  • MicroRNAs / genetics*
  • Prostatic Neoplasms / genetics*
  • Prostatic Neoplasms / metabolism
  • Proto-Oncogene Proteins c-pim-1 / chemistry
  • Proto-Oncogene Proteins c-pim-1 / genetics*
  • RNA Interference
  • RNA, Messenger / chemistry
  • RNA, Messenger / genetics
  • Radiation Tolerance / genetics*
  • Ribonuclease III / genetics
  • Ribonuclease III / metabolism

Substances

  • 3' Untranslated Regions
  • MIRN124 microRNA, human
  • MIRN144 microRNA, human
  • MicroRNAs
  • RNA, Messenger
  • PIM1 protein, human
  • Proto-Oncogene Proteins c-pim-1
  • Ribonuclease III