Synthesis and antileukemic activity of 1-[(quinolizidinylalkyl)amino]4/7-R-thioxanthen-9-ones

Farmaco. 1989 Nov;44(11):1069-82.

Abstract

Fifteen 1-(quinolizidinylalkyl)amino derivatives of thioxanthenone bearing different substituents on position 4 and 7 were prepared and tested in mice against lymphocytic leukemia P 388. These compounds were inactive or displayed only borderline activity (compounds 1, 10, 15).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / chemical synthesis*
  • Chemical Phenomena
  • Chemistry
  • Leukemia P388 / drug therapy*
  • Mice
  • Mice, Inbred Strains
  • Quinolizines / chemical synthesis*
  • Quinolizines / pharmacology
  • Spectrophotometry, Infrared
  • Spectrophotometry, Ultraviolet
  • Thioxanthenes / chemical synthesis*
  • Thioxanthenes / pharmacology

Substances

  • Antineoplastic Agents
  • Quinolizines
  • Thioxanthenes