Paeonol attenuates lipopolysaccharide-induced depressive-like behavior in mice

Psychiatry Res. 2016 Apr 30:238:116-121. doi: 10.1016/j.psychres.2016.02.033. Epub 2016 Feb 17.

Abstract

The present study was designed to detect the anti-depressant effects of paeonol and the possible mechanisms in the lipopolysaccharide-induced depressive-like behavior. Open-field test(OFT), tail suspension test(TST) and forced swimming test(FST) were used to evaluate the behavioral activity. The contents of 5-hydroxytryptamine (5-HT) and norepinephrine (NE) in mice hippocampus were determined by HPLC-ECD. Serum interleukin (IL)-1β, IL-6 and tumor necrosis factor (TNF)-α levels were evaluated by enzyme-linked immunosorbent assay (ELISA). Our results showed that LPS significantly decreased the levels of 5-HT and NE in the hippocampus. LPS also reduced open-field activity, as well as increased immobility duration in FST and TST. Paeonol administration could effectively reverse the alterations in the concentrations of 5-HT, NE and reduce the IL-6 and TNF-α levels. Moreover, paeonol effectively downregulated brain-derived neurotrophic factor (BDNF), tropomyosin-related kinase B (TrkB) and Nuclear factor-κB (NF-κB) in hippocampal. In conclusion, paeonol administration exhibited significant antidepressant-like effects in mice with LPS-induced depression.

Keywords: Inflammation; LPS-induced depression; Paeonol.

MeSH terms

  • Acetophenones / pharmacology*
  • Animals
  • Antidepressive Agents / pharmacology*
  • Brain-Derived Neurotrophic Factor / metabolism
  • Depression / chemically induced
  • Depression / drug therapy*
  • Depression / psychology
  • Depressive Disorder / drug therapy
  • Enzyme-Linked Immunosorbent Assay
  • Hindlimb Suspension
  • Hippocampus / drug effects
  • Interleukin-1beta / metabolism
  • Interleukin-6 / metabolism
  • Lipopolysaccharides
  • Male
  • Mice
  • Mice, Inbred ICR
  • NF-kappa B / metabolism
  • Norepinephrine / metabolism
  • Receptor, trkB / metabolism
  • Serotonin / metabolism
  • Signal Transduction / drug effects
  • Swimming
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Acetophenones
  • Antidepressive Agents
  • Brain-Derived Neurotrophic Factor
  • Interleukin-1beta
  • Interleukin-6
  • Lipopolysaccharides
  • NF-kappa B
  • Tumor Necrosis Factor-alpha
  • Serotonin
  • paeonol
  • Receptor, trkB
  • Norepinephrine