Curtius-like Rearrangement of an Iron-Nitrenoid Complex and Application in Biomimetic Synthesis of Bisindolylmethanes

Org Lett. 2016 May 6;18(9):2228-31. doi: 10.1021/acs.orglett.6b00864. Epub 2016 Apr 26.

Abstract

A Curtius-like rearrangement of hydroxamates to isocyanates was discovered. This reaction was initiated from an iron(II)-nitrenoid complex, which was generated by the iron(II)-catalyzed cleavage of N-O bonds of functionalized hydroxamates. To demonstrate the efficiency of this new Curtius-like rearrangement in synthetic chemistry, a biomimetic strategy for the one-pot preparation of bisindolylmethanes was developed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biomimetic Materials / chemical synthesis*
  • Biomimetic Materials / chemistry
  • Catalysis
  • Ferrous Compounds / chemistry*
  • Indoles / chemical synthesis*
  • Indoles / chemistry
  • Methane / analogs & derivatives
  • Methane / chemical synthesis*
  • Methane / chemistry
  • Molecular Structure

Substances

  • Ferrous Compounds
  • Indoles
  • Methane