Slug inhibits pancreatic cancer initiation by blocking Kras-induced acinar-ductal metaplasia

Sci Rep. 2016 Jul 1:6:29133. doi: 10.1038/srep29133.

Abstract

Cells in the pancreas that have undergone acinar-ductal metaplasia (ADM) can transform into premalignant cells that can eventually become cancerous. Although the epithelial-mesenchymal transition regulator Snail (Snai1) can cooperate with Kras in acinar cells to enhance ADM development, the contribution of Snail-related protein Slug (Snai2) to ADM development is not known. Thus, transgenic mice expressing Slug and Kras in acinar cells were generated. Surprisingly, Slug attenuated Kras-induced ADM development, ERK1/2 phosphorylation and proliferation. Co-expression of Slug with Kras also attenuated chronic pancreatitis-induced changes in ADM development and fibrosis. In addition, Slug attenuated TGF-α-induced acinar cell metaplasia to ductal structures and TGF-α-induced expression of ductal markers in ex vivo acinar explant cultures. Significantly, blocking the Rho-associated protein kinase ROCK1/2 in the ex vivo cultures induced expression of ductal markers and reversed the effects of Slug by inducing ductal structures. In addition, blocking ROCK1/2 activity in Slug-expressing Kras mice reversed the inhibitory effects of Slug on ADM, ERK1/2 phosphorylation, proliferation and fibrosis. Overall, these results increase our understanding of the role of Slug in ADM, an early event that can eventually lead to pancreatic cancer development.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Acinar Cells / pathology
  • Animals
  • Cell Transformation, Neoplastic / genetics
  • Disease Models, Animal
  • Epithelial-Mesenchymal Transition / genetics
  • Humans
  • Metaplasia / genetics*
  • Metaplasia / pathology
  • Mice
  • Mice, Transgenic
  • Pancreatic Ducts / metabolism
  • Pancreatic Ducts / pathology
  • Pancreatic Neoplasms / genetics*
  • Pancreatic Neoplasms / pathology
  • Pancreatitis, Chronic / genetics
  • Pancreatitis, Chronic / pathology
  • Proto-Oncogene Proteins p21(ras) / genetics*
  • Signal Transduction / genetics
  • Snail Family Transcription Factors / genetics*

Substances

  • Snai2 protein, mouse
  • Snail Family Transcription Factors
  • Hras protein, mouse
  • Proto-Oncogene Proteins p21(ras)