Tunable regulation of CREB DNA binding activity couples genotoxic stress response and metabolism

Nucleic Acids Res. 2016 Nov 16;44(20):9667-9680. doi: 10.1093/nar/gkw643. Epub 2016 Jul 18.

Abstract

cAMP response element binding protein (CREB) is a key regulator of glucose metabolism and synaptic plasticity that is canonically regulated through recruitment of transcriptional coactivators. Here we show that phosphorylation of CREB on a conserved cluster of Ser residues (the ATM/CK cluster) by the DNA damage-activated protein kinase ataxia-telangiectasia-mutated (ATM) and casein kinase1 (CK1) and casein kinase2 (CK2) positively and negatively regulates CREB-mediated transcription in a signal dependent manner. In response to genotoxic stress, phosphorylation of the ATM/CK cluster inhibited CREB-mediated gene expression, DNA binding activity and chromatin occupancy proportional to the number of modified Ser residues. Paradoxically, substoichiometric, ATM-independent, phosphorylation of the ATM/CK cluster potentiated bursts in CREB-mediated transcription by promoting recruitment of the CREB coactivator, cAMP-regulated transcriptional coactivators (CRTC2). Livers from mice expressing a non-phosphorylatable CREB allele failed to attenuate gluconeogenic genes in response to DNA damage or fully activate the same genes in response to glucagon. We propose that phosphorylation-dependent regulation of DNA binding activity evolved as a tunable mechanism to control CREB transcriptional output and promote metabolic homeostasis in response to rapidly changing environmental conditions.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Ataxia Telangiectasia Mutated Proteins / metabolism
  • Binding Sites
  • Cell Line
  • Cyclic AMP / metabolism
  • Cyclic AMP Response Element-Binding Protein / chemistry
  • Cyclic AMP Response Element-Binding Protein / genetics
  • Cyclic AMP Response Element-Binding Protein / metabolism*
  • DNA / genetics*
  • DNA / metabolism*
  • DNA Damage*
  • Energy Metabolism / genetics*
  • Gene Expression Regulation*
  • Gluconeogenesis / genetics
  • Male
  • Mice
  • Mice, Knockout
  • Phosphorylation
  • Protein Binding
  • Protein Interaction Domains and Motifs
  • Signal Transduction
  • Transcription Factors / metabolism

Substances

  • Crtc2 protein, mouse
  • Cyclic AMP Response Element-Binding Protein
  • Transcription Factors
  • DNA
  • Cyclic AMP
  • Ataxia Telangiectasia Mutated Proteins