[4 + 3] Cycloaddition of Phthalazinium Dicyanomethanides with Azoalkenes Formed in Situ: Synthesis of Triazepine Derivatives

J Org Chem. 2016 Sep 2;81(17):7597-603. doi: 10.1021/acs.joc.6b01296. Epub 2016 Aug 5.

Abstract

[4 + 3] cycloaddition of phthalazinium dicyanomethanides with in situ formed azoalkenes was achieved, providing an access to various 1,2,4-triazepine derivatives in moderate to excellent yields.

Publication types

  • Research Support, Non-U.S. Gov't