The polarity protein Scribble positions DLC3 at adherens junctions to regulate Rho signaling

J Cell Sci. 2016 Oct 1;129(19):3583-3596. doi: 10.1242/jcs.190074. Epub 2016 Aug 5.

Abstract

The spatial regulation of cellular Rho signaling by GAP proteins is still poorly understood. By performing mass spectrometry, we here identify the polarity protein Scribble as a scaffold for the RhoGAP protein DLC3 (also known as StarD8) at cell-cell adhesions. This mutually dependent interaction is mediated by the PDZ domains of Scribble and a PDZ ligand (PDZL) motif in DLC3. Both Scribble depletion and PDZL deletion abrogated DLC3 junctional localization. Using a RhoA biosensor and a targeted GAP domain, we demonstrate that DLC3 activity locally regulates RhoA-ROCK signaling at and Scribble localization to adherens junctions, and is required for their functional integrity. In a 3D model of cyst development, we furthermore show that DLC3 depletion impairs polarized morphogenesis, phenocopying the effects observed upon Scribble knockdown. We thus propose a new function for Scribble in Rho regulation that entails positioning of DLC3 GAP activity at cell junctions in polarized epithelial cells.

Keywords: Adherens junctions; Apical-basolateral polarity; PDZ domain interaction; Rho GTPase-activating protein; Tumor suppressor.

MeSH terms

  • Adherens Junctions / metabolism*
  • Caco-2 Cells
  • Cell Adhesion
  • Cell Polarity*
  • GTPase-Activating Proteins / metabolism*
  • Gene Knockdown Techniques
  • HEK293 Cells
  • Humans
  • Ligands
  • MCF-7 Cells
  • Membrane Proteins / chemistry
  • Membrane Proteins / metabolism*
  • PDZ Domains
  • Protein Binding
  • Signal Transduction*
  • Tumor Suppressor Proteins / chemistry
  • Tumor Suppressor Proteins / metabolism*
  • rho-Associated Kinases / metabolism
  • rhoA GTP-Binding Protein / metabolism

Substances

  • GTPase-Activating Proteins
  • Ligands
  • Membrane Proteins
  • SCRIB protein, human
  • STARD8 protein, human
  • Tumor Suppressor Proteins
  • rho GTPase-activating protein
  • rho-Associated Kinases
  • rhoA GTP-Binding Protein