Idebenone improves learning and memory impairment induced by cholinergic or serotonergic dysfunction in rats

Arch Gerontol Geriatr. 1989 May;8(3):225-39. doi: 10.1016/0167-4943(89)90005-8.

Abstract

The effects of idebenone, a cerebral metabolic enhancer, on learning and memory impairment in two rat models with central cholinergic or serotonergic dysfunction were investigated using positively reinforced learning tasks. A delayed alternation task using a T maze was employed to test the effect of idebenone on short-term memory impairment induced by a cholinergic antagonist, scopolamine. A correct response, defined as a turn toward the arm opposite to that in the forced run, was rewarded with food pellets. Scopolamine (0.2 and 0.5 mg/kg, i.p.) significantly decreased the correct responses to the chance level in the 60-s-delayed alternation task. The scopolamine (0.2 mg/kg, i.p.)-induced impairment of short-term memory was improved by idebenone (3-30 mg/kg, i.p.) or an acetylcholinesterase inhibitor, physostigmine (0.1 and 0.2 mg/kg, i.p.), administered simultaneously. The central serotonergic dysfunction model was produced by giving rats a diet deficient in tryptophan, a precursor of serotonin. The rats fed on a tryptophan-deficient diet (TDD) showed a slower learning process in the operant brightness discrimination task (mult V115 EXT) than did rats fed on a normal diet. Idebenone (60 mg/kg/day) admixed with the TDD decreased the number of lever-pressing responses emitted during the extinction periods. The percentage of correct responses was significantly higher in the idebenone-treated group than in the control TDD group. These results suggest that idebenone may improve both the impairment of short-term memory induced by a decreased cholinergic activity and the retardation of discrimination learning induced by central serotonergic dysfunction.

MeSH terms

  • Acetylcholine / physiology*
  • Animals
  • Benzoquinones*
  • Cerebral Cortex / drug effects
  • Cerebrovascular Disorders / complications*
  • Cerebrovascular Disorders / physiopathology*
  • Discrimination Learning / drug effects
  • Learning Disabilities / drug therapy*
  • Male
  • Memory Disorders / chemically induced
  • Memory Disorders / drug therapy*
  • Memory, Short-Term / drug effects
  • Quinones / administration & dosage
  • Quinones / pharmacology*
  • Rats
  • Rats, Inbred Strains
  • Scopolamine
  • Serotonin / physiology*
  • Ubiquinone / analogs & derivatives

Substances

  • Benzoquinones
  • Quinones
  • Ubiquinone
  • Serotonin
  • Scopolamine
  • idebenone
  • Acetylcholine