CDK5 functions as a tumor promoter in human colorectal cancer via modulating the ERK5-AP-1 axis

Cell Death Dis. 2016 Oct 13;7(10):e2415. doi: 10.1038/cddis.2016.333.

Abstract

Abnormal expression of cyclin-dependent kinase 5 (CDK5) has been found in several human cancers, whereas the role of CDK5 in the malignant development of colorectal cancer (CRC) has not been well characterized. Here we investigated the role of CDK5 in CRC and found that its expression was much higher in CRC tissues than that in normal tissues with a higher expression level of CDK5 closely correlating to advanced American Joint Committee on Cancer (AJCC) stage, poor differentiation, increased tumor size and poor prognosis of CRC. Biological function experiments showed that CDK5 regulated CRC cell proliferation and metastasis ability. Whole-genome microarray analysis, co-immunoprecipitation, in vitro kinase assay, western blotting, luciferase reporter assays and electrophoretic mobility shift assay (EMSA) showed that CDK5 could directly phosphorylate ERK5 at threonine (Thr) 732 and finally modulate the oncogenic ERK5-AP-1 axis. Further researches showed that CDK5-ERK5-AP-1 axis could promote progression of CRC carcinogenesis and had a significant correlation in human CRC samples. In summary, this study revealed the functional and mechanistic links between CDK5 and the oncogenic ERK5-AP-1 signaling pathway in the pathogenesis of CRC. These findings suggest that CDK5 has an important role in CRC development and may serve as a potential therapeutic target for CRC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing
  • Carcinogenesis / genetics
  • Carcinogenesis / pathology
  • Cell Cycle Proteins
  • Cell Line, Tumor
  • Cell Movement / genetics
  • Cell Proliferation / genetics
  • Colorectal Neoplasms / genetics
  • Colorectal Neoplasms / metabolism*
  • Colorectal Neoplasms / pathology*
  • Cyclin-Dependent Kinase 5 / metabolism*
  • Disease Progression
  • Down-Regulation / genetics
  • Female
  • Gene Expression Profiling
  • Gene Expression Regulation, Neoplastic
  • Gene Knockdown Techniques
  • Humans
  • Male
  • Middle Aged
  • Mitogen-Activated Protein Kinase 7 / metabolism*
  • Neoplasm Invasiveness
  • Neoplasm Metastasis
  • Phosphorylation
  • Phosphothreonine / metabolism
  • Signal Transduction*
  • Survival Analysis
  • Transcription Factor AP-1 / metabolism*
  • Up-Regulation / genetics

Substances

  • Adaptor Proteins, Signal Transducing
  • CDCA5 protein, human
  • Cell Cycle Proteins
  • Transcription Factor AP-1
  • Phosphothreonine
  • Cyclin-Dependent Kinase 5
  • CDK5 protein, human
  • MAPK7 protein, human
  • Mitogen-Activated Protein Kinase 7