[Binding of K-18 on the surface of tumor cells--flowcytometrical analysis in vitro]

Gan To Kagaku Ryoho. 1989 Aug;16(8 Pt 1):2627-31.
[Article in Japanese]

Abstract

After K-18 was contacted with various kinds of tumor cell lines in vitro, the binding pattern was examined. K-18 bound on the surface of K-562 cells showed the maximum levels 1 hr later and maintained the binding activity for 24 hrs in the analysis by flowcytometry. K-18 also bound to HeLa S3, KB, RPMI8226, P815, YAC-1 and L1210 cells. Fluorescent intensity on K-562 cells was stronger with whole molecules of K-18 than with F(ab')2 conjugated with melphalan. Normal human IgG could bind more on the surface of K-562 cells than F(ab')2 of IgG. These results suggest that K-18 might bind on tumor cells via IgG Fc receptors on their surface.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Antineoplastic Combined Chemotherapy Protocols / metabolism*
  • Cell Membrane / metabolism
  • Flow Cytometry
  • Humans
  • Immunoglobulin Fab Fragments / analysis
  • Immunoglobulin G / metabolism
  • Melphalan / metabolism
  • Rats
  • Receptors, Fc / metabolism
  • Tumor Cells, Cultured / metabolism*

Substances

  • Immunoglobulin Fab Fragments
  • Immunoglobulin G
  • Receptors, Fc
  • antineoplastic agent K 18
  • Melphalan